Ali Y, Alam MS, Hamid H, Husain A, Bano S, Dhulap A, Kharbanda C, Nazreen S, Haider S (2015) Design, synthesis and biological evaluation of piperic acid triazolyl derivatives as potent anti-inflammatory agents. Eur J Med Chem 92:490–500. https://doi.org/10.1016/j.ejmech.2015.01.001
Article CAS PubMed Google Scholar
Alotaibi F (2017) Design, synthesis and biological evaluation of novel estradiol-triazole analogs targeting epidermal growth factor receptors in colorectal cancer. Dissertation, South Dakota State University
Aneja B, Azam M, Alam S, Perwez A, Maguire R, Yadava U, Kavanagh K, Daniliuc CG, Rizvi MMA, Haq QMR (2018) Natural product-based 1, 2, 3-triazole/sulfonate analogues as potential chemotherapeutic agents for bacterial infections. ACS Omega 3:6912–6930. https://doi.org/10.1021/acsomega.8b00582
Article CAS PubMed PubMed Central Google Scholar
Banik BK, Banik I, Becker FF (2010) Asymmetric synthesis of anticancer β-lactams via staudinger reaction: utilization of chiral ketene from carbohydrate. Eur J Med Chem 45:846–848. https://doi.org/10.1016/j.ejmech.2009.11.024
Article CAS PubMed Google Scholar
Baraniak D, Kacprzak K, Celewicz L (2011) Synthesis of 3′-azido-3′-deoxythymidine (azt)—cinchona alkaloid conjugates via click chemistry: toward novel fluorescent markers and cytostatic agents. Bioorg Med Chem Lett 21:723–726. https://doi.org/10.1016/j.bmcl.2010.11.127
Article CAS PubMed Google Scholar
Bodnár B, Mernyák E, Wölfling J, Schneider G, Herman B, Szécsi M, Sinka I, Zupkó I, Kupihár Z, Kovács L (2016) Synthesis and biological evaluation of triazolyl 13α-estrone–nucleoside bioconjugates. Molecules 21:1212. https://doi.org/10.3390/molecules21091212
Article PubMed PubMed Central Google Scholar
Bonandi E, Christodoulou MS, Fumagalli G, Perdicchia D, Rastelli G, Passarella D (2017) The 1, 2, 3-triazole ring as a bioisostere in medicinal chemistry. Drug Discov Today 22:1572–1581. https://doi.org/10.1016/j.drudis.2017.05.014
Article CAS PubMed Google Scholar
Bori ID, Hung HY, Qian K, Chen CH, Morris-Natschke SL, Lee KH (2012) Anti-aids agents 88. Anti-hiv conjugates of betulin and betulinic acid with azt prepared via click chemistry. Tetrahedron Lett 53:1987–1989. https://doi.org/10.1016/j.tetlet.2012.02.022
Article CAS PubMed PubMed Central Google Scholar
Braje WM, Frackenpohl J, Schrake O, Wartchow R, Beil W, Hoffmann HMR (2000) Synthesis of 10,11-didehydro cinchona alkaloids and key derivatives. Helv Chim Acta 83:777–792. https://doi.org/10.1002/(SICI)1522-2675(20000412)83:4%3c777::AID-HLCA777%3e3.0.CO;2-W
Bunders C, Cavanagh J, Melander C (2011) Flustramine inspired synthesis and biological evaluation of pyrroloindoline triazole amides as novel inhibitors of bacterial biofilms. Org Biomol Chem 9:5476–5481. https://doi.org/10.1039/C1OB05605K
Article CAS PubMed PubMed Central Google Scholar
Caprioglio D, Torretta S, Ferrari M, Travelli C, Grolla AA, Condorelli F, Genazzani AA, Minassi A (2016) Triazole-curcuminoids: a new class of derivatives for “tuning” curcumin bioactivities? Bioorg Med Chem 24:140–152. https://doi.org/10.1016/j.bmc.2015.11.044
Article CAS PubMed Google Scholar
Carvalho AA, Galdino PM, Nascimento MV, Kato MJ, Valadares MC, Cunha LC, Costa EA (2010) Antinociceptive and antiinflammatory activities of grandisin extracted from virola surinamensis. Phytother Res 24:113–118. https://doi.org/10.1002/ptr.2882
Article CAS PubMed Google Scholar
Cassamale TB, Costa EC, Carvalho DB, Cassemiro NS, Tomazela CC, Marques M, Ojeda M, Matos MF, Albuquerque S, Arruda CC (2016) Synthesis and antitrypanosomastid activity of 1, 4-diaryl-1, 2, 3-triazole analogues of neolignans veraguensin, grandisin and machilin g. J Braz Chem Soc 27:1217–1228. https://doi.org/10.5935/0103-5053.20160017
Chandrashekhar M, Nayak VL, Ramakrishna S, Mallavadhani UV (2016) Novel triazole hybrids of myrrhanone c, a natural polypodane triterpene: synthesis, cytotoxic activity and cell based studies. Eur J Med Chem 114:293–307. https://doi.org/10.1016/j.ejmech.2016.03.013
Article CAS PubMed Google Scholar
Chen JK (2016) I only have eye for ewe: the discovery of cyclopamine and development of Hedgehog pathway-targeting drugs. Nat Prod Rep 33:595–601. https://doi.org/10.1039/c5np00153f
Article CAS PubMed PubMed Central Google Scholar
Chen X, McRae S, Parelkar S, Emrick T (2009) Polymeric phosphorylcholine− camptothecin conjugates prepared by controlled free radical polymerization and click chemistry. Bioconjug Chem 20:2331–2341. https://doi.org/10.1021/bc900339x
Article CAS PubMed Google Scholar
Cheng K, Liu J, Liu X, Li H, Sun H, Xie J (2009) Synthesis of glucoconjugates of oleanolic acid as inhibitors of glycogen phosphorylase. Carbohydr Res 344:841–850. https://doi.org/10.1016/j.carres.2009.02.012
Article CAS PubMed Google Scholar
Cheng K, Liu J, Sun H, Xie J (2010) Synthesis of oleanolic acid dimers as inhibitors of glycogen phosphorylase. Chem Biodivers 7:690–697. https://doi.org/10.1002/cbdv.200900086
Article CAS PubMed Google Scholar
Chu F, Zhang W, Guo W, Wang Z, Yang Y, Zhang X, Fang K, Yan M, Wang P, Lei H (2018) Oleanolic acid-amino acids derivatives: design, synthesis, and hepatoprotective evaluation in vitro and in vivo. Molecules 23:322. https://doi.org/10.3390/molecules23020322
Article CAS PubMed PubMed Central Google Scholar
Czyrski A, Resztak M, Świderski P, Brylak J, Główka FK (2021) The overview on the pharmacokinetic and pharmacodynamic interactions of triazoles. Pharmaceutics 13:1961. https://doi.org/10.3390/pharmaceutics13111961
Article CAS PubMed PubMed Central Google Scholar
Day JE, Sharp SY, Rowlands MG, Aherne W, Lewis W, Roe SM, Prodromou C, Pearl LH, Workman P, Moody CJ (2010) Inhibition of hsp90 with resorcylic acid macrolactones: synthesis and binding studies. Chem Eur J 16:10366–10372. https://doi.org/10.1002/chem.201001119
Article CAS PubMed Google Scholar
Dheer D, Singh V, Shankar R (2017) Medicinal attributes of 1, 2, 3-triazoles: current developments. Bioorg Chem 71:30–54. https://doi.org/10.1016/j.bioorg.2017.01.010
Article CAS PubMed Google Scholar
Dhyani MV, Satpati D, Korde A, Sarma HD, Kumar C, Banerjee S (2010) Preparation and preliminary bioevaluation of 99mtc (co) 3–11β-progesterone derivative prepared via click chemistry route. Nucl Med Biol 37:997–1004. https://doi.org/10.1016/j.nucmedbio.2010.04.003
Article CAS PubMed Google Scholar
Ding C, Zhang Y, Chen H, Wild C, Wang T, White MA, Shen Q, Zhou J (2013) Overcoming synthetic challenges of oridonin a-ring structural diversification: regio-and stereoselective installation of azides and 1, 2, 3-triazoles at the C-1, C-2, or C-3 position. Org Lett 15:3718–3721. https://doi.org/10.1021/ol401618c
Article CAS PubMed PubMed Central Google Scholar
Dirks M (2021) Bioactivity assessment of veratrum californicum alkaloids. Dissertation, Boise State University
Dreier I, Hansen LH, Nielsen P, Vester B (2014) A click chemistry approach to pleuromutilin derivatives. Part 3: extended footprinting analysis and excellent mrsa inhibition for a derivative with an adenine phenyl side chain. Bioorg Med Chem Lett 24:1043–1046. https://doi.org/10.1016/j.bmcl.2014.01.019
Article CAS PubMed Google Scholar
Dreier I, Kumar S, Søndergaard H, Rasmussen ML, Hansen LH, List NH, Kongsted J, Vester B, Nielsen P (2012) A click chemistry approach to pleuromutilin derivatives, part 2: conjugates with acyclic nucleosides and their ribosomal binding and antibacterial activity. J Med Chem 55:2067–2077. https://doi.org/10.1021/jm201266b
Article CAS PubMed Google Scholar
Dupuis SN, Robertson AW, Veinot T, Monro SM, Douglas SE, Syvitski RT, Goralski KB, McFarland SA, Jakeman DL (2012) Synthetic diversification of natural products: semi-synthesis and evaluation of triazole jadomycins. Chem Sci 3:1640–1644. https://doi.org/10.1039/C2SC00663D
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